HETEROCYCLES
An International Journal for Reviews and Communications in Heterocyclic ChemistryWeb Edition ISSN: 1881-0942
Published online by The Japan Institute of Heterocyclic Chemistry
Regular Issue
Vol. 14, No. 1, 1980
Published online:
■ Stereo- and Regio-selective Formation of Telomers of 2-Oxazolone with Polyhalomerhanes (Structure and Reactivity)
Yoshihiro Abe* and Takehisa Kunieda
*Faculty of Pharmaceutical Sciences, University of Tokyo, Hongo, Bunkyo-ku, Tokyo 113, Japan
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■ Stereospecific S-Assisted Cationic Cyclization. A Synthetic Application to Thiasteroids
Tadao Terasawa* and Toshihiko Okada
*Shionogi Research Laboratories, Shionogi & Co. Ltd., Fukushima-ku, Osaka 553-0002, Japan
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■ Synthetic Applications of Reactions of N-Substituted Pyrroles and Indoles with Palladium Acetate
Toshio Itahara*
*Department of Bioengineering, Faculty of Engineering, Kagoshima University, Korimoto, Kagoshima 890-0065, Japan
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■ One Step Synthesis of 4-Substituted Indoles
Masanori Somei,* Fumio Yamada, and Chikara Kaneko
*Faculty of Pharmaceutical Sciences, Kanazawa University, 13-1 Takara-machi, Kanazawa 920-0934, Japan
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■ Five-Step Synthesis of 4-Alkylindoles
Mitsutaka Natsume* and Hideaki Muratake
*Research Foundation Itsuu Laboratory, 2-28-10 Tamagawa, Setagaya-ku, Tokyo 158, Japan
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■ Synthesis and Cycloaddition Reactions of 3-Cyanoindolizines
Kiyoshi Matsumoto,* Yukio Ikemi-Kono, Takane Uchida, and Leo A. Paquette
*College of Liberal Arts and Science, Kyoto University, Yoshida, Sakyou-ku, Kyoto 606-8501, Japan
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■ Syntheses of Indolizine Derivatives and Their Reactions
Keiji Kurata, Yasushi Tajima, Hiroyoshi Awaya, Yoshinori Tominaga, Yoshiro Matsuda, and Goro Kobayashi*
*Faculty of Pharmaceutical Sciences, Nagasaki University, 1-14, Bunkyo-machi, Nagasaki 852-8521, Japan
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■ Convenient Synthesis of Pyranoindolizines
Akikazu Kakehi,* Suketaka Ito, Kazunori Nakanishi, Kozo Watanabe, and Masahiko Kitagawa
*Department of Chemistry and Material Engineering, Faculty of Engineering, Shinshu University, 4-17-1 Wakasato, Nagano 380-8553, Japan
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■ Heterocycle Syntheses Using o-Lithiomethylphenyl Isocyanide Intermediates
Yoshihiko Ito,* Kazuhiro Kobayashi, Norihiko Seko, Masayuki Maeno, and Takeo Saegusa
*Department of Synthetic Chemistry, Faculty of Pharmaceutical Sciences, Kyoto University, Yoshida, Sakyou-ku, Kyoto 606-8501, Japan
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■ Synthesis of 3-Acetyl and 3-Aroyl-1,2-benzisoxazole Derivatives
Teruo Yamamori* and Ikuo Adachi
*Shionogi Research Laboratories, Shionogi & Co. Ltd., Fukushima-ku, Osaka 553-0002, Japan
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■ Heterocycles from Acylation of Some Imines with Pyridinecarbonyl Chlorides
Takeaki Naito,* Okiko Miyata, and Ichiya Ninomiya
*Kobe Women’s College of Pharmacy, Motoyamakita, Higashinad, Kobe, Hyogo 658, Japan
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■ Reaction of Dichlorocarbene to Pyridines and Condensed Pyridines
Yoshiki Hamada* and Michiharu Suigura
*Faculty of Pharmacy, Meijo University, 150 Yagotoyama, Tenpaku, Nagoya 468-8503, Japan
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■ New Alkylations of Quinoline N-Oxides
Fuminori Sato, Masayoshi Yamashita, Makoto Nishikawa, Hiroshi Noda, Seitaro Saeki, and Masatomo Hamana*
*Faculty of Pharmaceutical Sciences, Kyushu University, 3-1-1 Maidashi, Higashi-ku, Fukuoka 812-8582, Japan
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■ Diels-Alder Reaction of 1-Methyl-4-substituted 2(1H)-Pyridones with Alkyl-1,3-butadiene. A Novel Synthesis of Isoquinoline Derivatives
Hiroshi Tomisawa,* Reiko Fujita, Hideki Kato, and Hiroshi Hongo
*Tohoku Pharmaceutical University, 4-4-1 Komatsushima, Aoba-ku, Sendai 981-8558, Japan
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■ The Reaction of 1-Substituted 3,5-Dinitro-4-pyridones with Primary Amines
Eizo Matsumura,* Masahiro Ariga, Yasuo Tohda, and Hiroaki Oka
*Department of Chemistry, Osaka Kyoiku University, 4-698-1 Asahigaoka, Kashiwara, Osaka 582-8582, Japan
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■ Synthesis of Large Memberd Heterocycles by Regioselective Remote Photocyclization. Photoreaction of Sulfide-containing Phthalimides
Yasuhiko Sato,* Masao Wada, Hideo Nakai, Yasumaru Hatanaka, and Yuichi Kanaoka
*Organic Chemistry Research Laboratory, Tanabe Seiyaku Co.Ltd., 2-2-50, Kawagishi, Toddda, Saitama 335-8505, Japan
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■ Photochemistry of Conjugated Nitrogen-carbonyl Systems. Photoaddition Reaction of Hydroxylazobenzenes and the Related Thione Analogs with Olefins
Yuichi Kanaoka,* Masato Hasebe, and Eisuke Sato
*Faculty of Pharmaceutical Sciences, Hokkaido University, Kita 12 Nishi 6, Kita-ku, Sapporo, Hokkaido 060-0812, Japan
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■ Photochemical Addition of 6-Cyano-1,3-dimethyluracil to Substituted Acetylenes and Olefins
Isao Saito,* Koji Shimozono, and Teruo Matsuura
*Department of Synthetic Chemistry, Faculty of Pharmaceutical Sciences, Kyoto University, Yoshida, Sakyou-ku, Kyoto 606-8501, Japan
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■ Synthesis and Related Reactions of 5- and 10-Thiaisoalloxazines
Yoshifumi Maki,* Mikio Suzuki, Tokiyuki Hiramitsu, Keiji Kameyama, and Ko Tanabe
*Gifu Pharmaceutical University, 6-1 Mitahora-higashi 5-chome, Gifu 502-8585, Japan
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■ Studies on the 3-Substituted 3H-1,2,3-Triazolo[4,5-d]pyrimidines
Takeo Higashino,* Eisaku Hayashi, and Tatsuhiko Katori
*Shizuoka College of Pharmacy, 2-2-1, Oshika, Shizuoka-shi, 442 Shizuoka, Japan
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■ On 6-C-Substituted Purine and 9-β-D-Ribofuranosylpurine Derivatives: Synthesis of 6-Dicyanomethylpurines and 3-Amino-2-(purin-6-yl)acrylonitriles
Tadashi Miyasaka,* Norimitsu Hamamichi, and Hiroshi Suemune
*School of Pharmaceutical Sciences, Showa University, 1-5-8 Hatanodai, Shinagawa-ku, Tokyo 142-8555, Japan
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■ Homolytic Carbon-Carbon Bond Formation on Pyrimidine Derivatives
Takao Sakamoto,* Takeji Sakasai, Takayasu Ono, and Hiroshi Yamanaka
*Graduate School of Pharmaceutical Sciences, Tohoku University, Aramaki, Aoba-ku, sendai 980-8578, Japan
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■ On the Reduction of 2(1H)-Pyrimidinones with Sodium Borohydride
Choji Kashima,* Yuko Yokota, Takehiko Nishio, and Akira Katoh
*Department of Chemistry, University of Tsukuba, 1-1-1 Ten-nodai, Tsukuba-shi, Ibaraki, 305-8571, Japan
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■ Heterocycles from Peptido-aminobenzophenone Derivatives
Kentaro Hirai,* Teruyuki Ishiba, Hirohiko Sugimoto, and Toshio Fujishita
*Shionogi Research Laboratories, Shionogi & Co. Ltd., Fukushima-ku, Osaka 553-0002, Japan
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■ Syntheses of Apogalanthamine Analogs as α-Adrenergic Blocking Agents
Shigeru Kobayashi,* Masaru Kihara, Yukio Ishida, and Tetsuro Shingu
*Faculty of Pharmaceutical Sciences, University of Tokushima, Sho-machi, Tokushima 770-8505, Japan
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■ Ring Transformation of Indoles: Synthesis of 1H-1-Benzazepines
Masazumi Ikeda,* Toshiko Uno, Kazunori Ohno, and Yasumitsu Tamura
*Kyoto Pharmaceutical University, Misasagi-Shichonocho, Yamashina, Kyoto 607-8414, Japan
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■ Syntheses of Nitrogen-containing Heterocyclic Compounds by the Use of Cyclopropenium Salt
Shigeo Yoneda, Hideo Hirai, Yoshio Katsuro, and Zen-ichi Yoshida*
*Faculty of Engineering, Kyoto University, Yoshida, Sakyou-ku, Kyoto 606-8501, Japan
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■ Synthesis of Pyrroles, Pyridines, and Azepines from 2H-Azirines
Masumi Saruwatari, Sumiko Hatano, Kazuaki Isomura, and Hiroshi Taniguchi*
*Research Institute of Industrial Science, Faculty of Engineering, Kyushu University, 6-1, Kasuga-koen, Kasuga 816-8580, Japan
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■ Synthesis of Seven-membered Heterocycles Containing Fluoroalkyl Groups
Masamichi Maruta, Satoshi Kubota, Norihiko Yoshimura, Tomoya Kitazume, and Nobuo Ishikawa*
*Department of Chemical Technology, Faculty of Engineering, Tokyo Institute of Technology, 2-12-1,Oh-Okayama, Meguro-ku, Tokyo 152-8552, Japan
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■ Photosensitized Oxygenation of 1,3-Oxazepines
Akihiko Tokida, Keiji Okada, and Toshio Mukai*
*Department of Chemistry, Faculty of Science, Tohoku University, Aoba-ku, Ssendai 980-8578, Japan