HETEROCYCLES
An International Journal for Reviews and Communications in Heterocyclic ChemistryWeb Edition ISSN: 1881-0942
Published online by The Japan Institute of Heterocyclic Chemistry
Regular Issue
Vol. 20, No. 1, 1983
Published online:
■ Synthetic Studies on Some Thiamodified Adamantane Skeletons
Tadashi Sasaki, Shoji Eguchi, Shinichi Yamada, and Hiroshi Ban
*Faculty of Engineering, Nagoya Institute of Technology, Gokiso-cho, Showa-ku, Nagoya 466-8555, Japan
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■ Thioamide-Claisen Rearrangements and Its Application to the Syntheses of Indole Alkaloids
Seiichi Takano, Michiyasu Hirama, and Kunio Ogasawara
*Pharmaceutical Institute, Tohoku University, Aobayama, Sendai 980-8578, Japan
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■ A New Method for the Preparation of 3,4-Dihydro-β-carbolines via Alkylthioiminium Salt
Akihiko Ishida, Tohru Nakamura, Kunihiko Irie, and Tokuro Oh-ishi
*Discovery Research Laboratory, Tanabe Seiyaka, 2-2-50, Kawagishi, Toddda, Saitama 335-8505, Japan
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■ Synthesis of (±)-Lupinine and (±)-Epilupinine Utilizing the Anodic Oxidation of Lactams
Makoto Okita, Takeshi Wakamatsu, and Yoshio Ban
*Faculty of Pharmaceutical Sciences, Toho University, 2-2-1, Miyama, Funabashi, Chiba 274-8510, Japan
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■ A Novel Highly Selective Chiral Induntion Utilizing a Functional Heterocyclic Compound, 4(R)-MCTT
Yoshimitsu Nagao, Takehisa Inoue, Takao Ikeda, Eiichi Fujita, and Shunji Terada
*Institute for Chemical Research, Kyoto University, Uji, Kyoto 611-0011, Japan
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■ Studies Directed towards Total Synthesis of Saframycin [I]
Hideshi Kurihara and Hiroshi Mishima
*Fermentation Research Laboratories, Sankyo Co., Ltd., 1-2-58 Hiromachi, Shinagawa-ku, Tokyo 140-8710, Japan
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■ Dioxopyrroline, an Ambident Dienophile in Diels-Alder Reaction
Yoshisuke Tsuda, Takeshi Oshima, Takehiro Sano, and Jun Toda
*Faculty of Pharmaceutical Scicences, Kanazawa University, 13-1 Takara-machi, Kanazawa 920-0934, Japan
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■ Syntheses of Biologically Active 4-Aryl-1,2,3,4-tetrahydroisoquinoline Derivatives under Control of the Orientation of Polonovski Rreaction
Takashi Nomoto, Nobuyuki Nasui, and Hiroaki Takayama
*Faculty of Pharmaceutical Sciences, Teikyo University, 1091-1 Suarashi, Sagamiko-machi, Tsukui-gun, Kanagawa 199-0195, Japan
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■ Application of an Oxygenative Nucleophile Introduction Reaction to 2-Alkynyl-1,2-dihydropyridine Derivatives
Masashi Ogawa and Mitsutaka Natsume
*Research Foundation Itsuu Laboratory, 2-28-10 Tamagawa, Setagaya-ku, Tokyo 158, Japan
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■ Synthetic Studies on the Polyether Antibiotics (Part 1). A New Method for the Synthesis of Functionalized Tertahydrofurans and Tetrahydropyrans
Yuji Oikawa, Kiyoshi Horita, and Osamu Yonemitsu
*Faculty of Pharmaceutical Sciences, Hokkaido University, Kita 12 Nishi 6, Kita-ku, Sapporo, Hokkaido 060-0812, Japan
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■ Asymmetric Synthesis of (+)-Thienamycin
Masakatsu Shibasaki, Atsushi Nishida, and Shiro Ikegami
*Faculty of Pharmaceutical Sciences, Teikyo University, 1091-1, Sagamiko, Kanagawa 199-0195, Japan
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■ Synthesis of Heterocyclic Compounds by the Sulfeno-cycloamination and Its Application to Natural Products Synthesis
Masataka Ihara, Tatsushi Ohsawa, Keiichiro Fukumoto, and Tetsuji Kametani
*Graduate School of Pharmaceutical Sciences, Tohoku University, Aramaki, Aoba-ku, sendai 980-8578, Japan
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■ Oxidative Dimerization of Tryptophan Derivatives. Total Synthesis of Ditryphenaline and Folicanthine
Masako Nakagawa, Hioryuki Sugumi, Shinichi Kodato, and Tohru Hino
*Faculty of Pharmaceutical Sciences, Chiba University, 1-33 Yayoi-cho, Inage-ku, Chiba 263-8522, Japan
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■ Synthesis of Heterocycles Using Isothiocyanatomethanide
Yoshiki Ohshiro, Ken-ichiro Hayashi, Atsushi Yamada, Gen-ichi Ishibashi, Toshikazu Hirao, and Toshio Agawa
*Department of Applied Chemistry, Faculty of Engineering, Osaka University, 2-1 Yamadaoka, Toyonaka, Osaka 560-0043, Japan
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■ Reactions of Pyridone Derivatives with Isocyanates; A Simple Preparation of 1,3,5-Triazine Derivatives
Yoshiro Furukawa, Masami Sawada, Yoshio Takai, and Terukiyo Hanafusa
*The Institute of Scientific and Industrial Research, Osaka University, 8-1. Mihogaoka, Ibaraki, Osaka 567-0047, Japan
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■ Ruthenium Tetroxide Oxidation of N-Alkyl-lactams
Yukimi Takai, Shigeyuki Yoshifuji and Yoshihiro Nitta
*School of Pharmacy, Hokuriku University, 3-Ho, Kanagawa machi, Kanazawa 920-1181, Japan
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■ Novel Cage Compounds from the Reaction of Thiazolium N-Methylide with Methylenecyclopropene
Otohiko Tsuge, Shuji Kanemasa, Hiroshi Shimoharada, and Shigeori Takenaka
*Research Institute of Industrial Science, Faculty of Engineering, Kyushu University, 6-1, Kasuga-koen, Kasuga 816-8580, Japan
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■ Selective Methylation of Intramolecular N and S Groups — Possible Formation of σ-Ammoniosulfuranes —
Kin-ya Akiba, Kohichi Takee, Katsuo Ohkata, Yoshio Ohara, and Naoki Inamoto
*Department of Chemistry, Faculty of Science, Hiroshima University, 1-3-1 Kagamiyama, Higashi-Hiroshima, Hiroshima 739-8526, Japan
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■ The Phoyochemistry of Annulenylion-Annulenone Cycle as a Model of Bacteriorhodospin
Haru Ogawa, Tadashi Inoue, Taiji Imoto, Hidefumi Kato, and Yoichi Taniguchi
*Faculty of Pharmaceutical Sciences, Kyushu University, 3-1-1 Maidashi, Higashi-ku, Fukuoka 812-8582, Japan
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■ Thiacrown Ethers and Derivatives: Preparation and Applications for Organic Reactions
Naomichi Furukawa, Koji Imaoka, and Shigeru Oae
*Department of Chemistry, University of Tsukuba, 1-1-1 Ten-nodai, Tsukuba-shi, Ibaraki, 305-8571, Japan
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■ Reagent Design and Study of 1,4-Dithiin as Promising Class of Reagents (Synthons) for Cycloadditioon. The Diels-Alder Reactions with Anthracene Derivatives via Charge-transfer Complexes
Kenji Hayakawa, Nobuko Mibu, Eiji Osawa, and Ken Kanematsu
*Faculty of Pharmaceutical Sciences, Kyushu University, 3-1-1 Maidashi, Higashi-ku, Fukuoka 812-8582, Japan
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■ Azulenophane VIII. Conformations of Dithia[3.3]azulenophanes
Yoshimasa Fukazawa, Jun Tsuchiya, Masao Sobukawa, and Sho Ito
*Department of Chemistry, Faculty of Science, Hiroshima University, 1-3-1 Kagamiyama, Higashi-Hiroshima, Hiroshima 739-8526, Japan
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■ Heterocycles Synthesis of Electrophilic Addition to Acetylenes
Shinjiro Kobayashi, Muneyuki Mastumoto, and Hiroshi Taniguchi
*Department of Applied Chemistry, Faculty of Engineering, Kyushu University, 6-10-1 Hakozaki, Higashi-ku, Fukuoka 812-8581, Japan
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■ Synthesis of Furans and Butenolides Using Acylketene Dithioacetals
Yoshio Negishi, Renji Okazaki, and Naoki Inamoto
*Department of Chemistry, Scool of Science, University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo 113-0033
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■ Formation and Reactivity of Dilithiated N-Acylfurfurylamines
Kosei Ohno and Minoru Machida
*Faculty of Pharmaceutical Scicences, Higashinihonngakuen University, 1757 Kanazawa, Toubetu-cho, Ishikari-gun, Hokkaodo 061-0212, Japan
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■ Synthesis of Some Nitrogen Heterocycles Using Diketene-Acetone Adduct
Masayuki Sato, Hiromichi Ogasawara, Norio Kanuma, Keiko Kato, Eriko Yoshizumi, Masako Sakai, and Tetsuzo Kato
*Pharmaceutical Institute, Tohoku University, Aobayama, Sendai 980-8578, Japan
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■ Synthesis and Properties of 1,3-Thiazinones
Yutaka Yamamoto and Shuhei Ohnishi
*Faculty of Pharmaceutical Sciences, Tohoku Pharmaceutical University, 4-4-1 Komatsushima, Aoba-ku, Sendai 981-8558, Japan
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■ Synthesis of 3-Substituted 1,2,4-Triazines
Masaaki Yokoyama, Etsuko Takaharu, Yuichi Aizawa, Shoetsu Konno, and Hiroshi Yamanaka
*Pharmaceutical Institute, Tohoku University, Aobayama, Sendai 980-8578, Japan
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■ Introduction of C-Substituents into the Pyrazine Ring
Akihiro Ohta, Yasuo Akita, and Masami Inoue
*Tokyo University of Pharmacy and Life Science, 1432-1 Horinouchi, Hachioji, Tokyo 192-0392, Japan
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■ A New Procedure for the Introduction of an Amino Group to Azaheterocycles
Hiroshi Hara and Henk C. van der Plas
*Laboratory of Organic Chemistry, Agricultural University, De Dreijen 5, 6703 BC Wageningen, The Netherlands