HETEROCYCLES
An International Journal for Reviews and Communications in Heterocyclic ChemistryWeb Edition ISSN: 1881-0942
Published online by The Japan Institute of Heterocyclic Chemistry
Special Issue
Special Issues of the 19th International Congress of Heterocyclic Chemistry's Special Issues, Vol. 21, No. 2, 1984
Published online:
■ Naturally Occurring Bioactive Benzo[de]-1,6-naphthyridines from the Sea Sponge Aaptos aaptos
Hideshi Nakamura, Jun’ichi Kobayashi, Reiko Abe, Yasushi Ohizumi, and Yoshimasa Hirata
*Institute of Life Science, Mitsubishi Kasei, Minaiooya-11, machida-shi, Tokyo 194
Published online:
■ Synthesis and Antihypertensive Activity of Some Fused Quinazoline Derivatives
Kang-Chien Liu and Ji-Wang Chern
*School of Pharmacy, National Defense Medical Center, P.O. Box 90048-508, Neihu, Taipei, Taiwan, R.O.C.
Published online:
■ Synthesis of New Benzopyrano/4,3-b/pyridine Ring Systems
J. Bálint, M. Rákosi, Zs. Szegény, and R. Bognár
*BIOGAL Pharmaceutical Works, H-4042 Debrecen, Hungary
Published online:
■ Synthesis of 4-Deoxy-4-C-ethylphosphinyl-D-ribo-and -L-lyxo-furanoses
Y. Nakamura, H. Yamamoto, S. Inokawa, and M. Yamashita
*Department of Chemistry, Faculty of Science, Okayama University, 3-1-1 Tsushima-naka, Okayama 700-8530, Japan
Published online:
■ Synthesis of L-Idopyranose Derivatives Having a Phosphorus Atom in the Hemiacetal Ring
Mitsuji Yamashita, Manabu Yamada, Kenji Tsunekawa, Tatsuo Oshikawa, and Saburo Inokawa
*Department of Applied Chemistry, Faculty of Engineering, Shizuoka University, 3-5-1 Johoku, Hamamatsu 432-8561, Shizuoka, Japan
Published online:
■ Synthesis of Tunicaminyl Uracil
Tetsuo Suami, Hiroaki Sasai, and Kazuhiro Matsuno
*The Institute of Scientific and Industrial Research, Osaka University, 8-1, Mihogaoka, Ibaraki, Osaka 567-0047, Japan
Published online:
■ Nin-Mesitylene-2-sulfonylyryptophan, a New Tryptophan Derivative, and Its Application for Peptide Synthesis
Nobutaka Fujii, Shiro Futaki, Kouichi Yasumura, Kenichi Akaji, and Haruaki Yajima
*Graduate School of Pharmaceutical Sciences, Kyoto University, 46-29 Yoshida-shimoadachi-machi, Sakyo-ku, Kyoto 606-8501, Japan
Published online:
■ Chemistry of Nucleoside-Amino Acid Adducts and Its Relevance to Photoinduced Lesions
Isao Saito, Hiroshi Sugiyama, M. B. Gupta, and Teruo Matsuura
*Department of Synthetic Chemistry, Faculty of Pharmaceutical Sciences, Kyoto University, Yoshida, Sakyou-ku, Kyoto 606-8501, Japan
Published online:
■ Unconventional Toxic Heterocycles of Clitocybe acromelalga
Katsuhiro Konno, Haruhisa Shirahama, and Takeshi Matsumoto
*Faculty of Science, Hokkaido University, Kita 10 Nishi 8, Kita-ku, Sapporo, Hokkaido 060-0810, Japan
Published online:
■ Synthesis of Quinazolines and 1,4-Benzodiazepines
Jan Bergman, Anna Brynolf, and Björn Elman
*Department of Organic Chemistry, Royal Institute of Technology, SE-100 44 Stockholm, Sweden
Published online:
■ Preparation and Reactions of 3-Benzoyl-3,4-dihydro-4-quinazolinecarbonitrile (Quinazoline Reissert Compound)
Takeo Higashino, Hiroyasu Kokubo, and Eisaku Hayashi
*Shizuoka College of Pharmacy, 2-2-1, Oshika, Shizuoka-shi, 442 Shizuoka, Japan
Published online:
■ Novel Mesoionic Heterocycles
Willy Friedrichsen, Andreas Böttcher, Tony Debaerdemaeker, Gisela Möckel, and Martha Schildberg
*Institut für Organische Chemie, Universität Kiel, Olshausenstrasse. 40, D-24098 Kiel, Germany
Published online:
■ The Reaction of 5-Benzalimino-1,2,4-triazoles with Substituted Acetyl Chlorides
József Reiter, László Pongó, Pál Sohár, and Péter Dvortsák
*EGIS Pharmaceuticals Ltd.,, H-1475 Budapest P.O.B. 100, Hungary
Published online:
■ Palladium Catalyzed Polyhetero-Claisen Rearrangement of 3-Allylthio-1,2,4-triazin-5(2H)-ones
Masato Mizutani, Yuzuru Sanemitsu, Yoshinao Tamaru, and Zen-ichi Yoshida
*Research Department, Sumitomo Chemical Co. Ltd., 4-2-1, Takatsukasa, Takarazuka, Hyogo, Japan
Published online:
■ A New, Synchronous Construction of Some Fused Pyrimidines by the Reaction of 6-Arylidenehydrazino-1,3-dimethyluracils with Thionyl Chloride
Misuzu Ichiba, Sadao Nishigaki, and Kentaro Senga
*Pharmaceutical Institute, School of Medicine, Keio University, Shinanomachi 35, Shinjuku, Tokyo 160-0016, Japan
Published online:
■ 1,3-Dipolar Cycloaddition Reactions of Thiazolo[5,4-d]pyrimidine 1-Oxides and Thiazolo[4,5-g]quinazoline 1-Oxides with Acetylenic Esters
Keitaro Senga, Misuzu Ichiba, Hashime Kanazawa, and Sadao Nishigaki
*Pharmaceutical Institute, School of Medicine, Keio University, Shinanomachi 35, Shinjuku, Tokyo 160-0016, Japan
Published online:
■ 4-Dicyanomethylene-1,4-dihydropyrimidines and Pyrido[4,3-d]pyrimisine-8-carbonitriles from Enaminonitoriles
Hans Junek and Martin Mittelbach
*Institute for Organic Chemistry, Karl-Franzens-University Graz, Heinrichstrasse. 28, A-8010 Graz, Austria
Published online:
■ Heterocyclic Syntheses with Brominated Malononitriles
Robert W. Morrison, Jr. and W. Revill Mallory
*Wellcome Research Laboratories, Burroughs Wellcome Co., 3030 Cornwallis Road, Research Triangle Park, NC 27709, U.S.A.
Published online:
■ Synthesis of 1,2,4-Triazino[6,5-e]1,2,4-triazines, 1,2,4-Triazino[6,5-e]1,2,4-thiadiazines and 1,2,4-Triazino[5,6-e]1,2,4-thiadiazines
Hans Neunhoeffer and Heinz Hammann
*Institut für Organische Chemie, Technische Hochschule Darmstadt, Petersenstrasse, 22 D-6100 Darmstadt, Germany
Published online:
■ Synthesis of 6-Hydroxy-4-(2’-di-n-propylaminoethyl)indole
Teresa Lee and Joseph G. Cannon
*Division of Medicinal and Natural Products Chemistry, College of Pharmacy, University of Iowa, Iowa City, Iowa 52242, U.S.A.
Published online:
■ Regioselective Vinylation of Indoles with Olefins and PdCl2
Yasuoki Murakami, Yuusaku Yokoyama, and Tsuyoshi Aoki
*School of Pharmaceutical Sciences, Toho University, 2-2-1, Miyama, Funabashi, Chiba 274-8510, Japan
Published online:
■ A New Versatile Synthesis of 4-Nitroindoles
Jan Bergman, Peter J. O. Sand, and Ulf Tilstam
*Department of Organic Chemistry, Royal Institute of Technology, SE-100 44 Stockholm, Sweden
Published online:
■ Reactions of Ethyl Phenylpropiolate with Indole Derivatives
M. Y. Shandala, H. A. Khatab, and N. Y. Yahya
*Department of Chemistry, College of Science, University of Mosul, Mosul, Iraq
Published online:
■ A Novel Spiro System: 2-Oxo-1’,2’,4’,5’-tetrahydro-spiro[3H-indole-3,3’-1,2,4,5-tetrazune]-6’-thione
Krishna C. Joshi, Pooran Chand, and Anshu Dandia
*Department of Chemistry, University of Rajasthan, Jaipur 302 004, India
Published online:
■ A Novel Spiro System: 4’,7’-Dihydro-8’-phenyl-spiro{3H-indole-3,6’-[pyrazolo(3,2-d)-1,3,5-thiadiazepine]}-2,3’(1H) Dione
Krishna C. Joshi, Pooran Chand, and Anshu Dandia
*Department of Chemistry, University of Rajasthan, Jaipur 302 004, India
Published online:
■ Tetrahydro-β-carboline- and β-Carboline-3-carboxamides
R. T. Coutts, R. G. Micetich, R. A. Locock, G. B. Baker, A. Benderley, J. Pyrozko, T. W. Hall, and T. Dewhurst
*Faculty of Pharmacy and Pharmaceutical Sciences, University of Alberta, Edmonton, Alberta, T6G 2G2, Canada
Published online:
■ Reactions of Haloketenes with Ethyl N-(2-Pyridyl)formimidates and 2-Arylideneaminopyridines
Nobuya Katagiri, Ryuji Niwa, and Tetsuzo Kato
*Pharmaceutical Institute, Tohoku University, Aobayama, Sendai 980-8578, Japan
Published online:
■ Photochemical Formation and Transznnlar Reactions of Medium-sized Nitrogen Heterocycles
Tuvia Sheradsky and Reuven Moshenberg
*Department of Organic Chemistry, The Hebrew University of Jerusalem, Jerusalem 91904, Israel
Published online:
■ 4-Diazomethylcoumarins as Stable Diazoalkanes. Their Facile Isomerization into Benzopyrano[3,4-c]pyrazol-4(3H)-ones
Keiichi Ito, Kazuo Nagasawa, and Junko Maruyama
*Hokkaido College of Pharmacy, 7-1 Katsuraoka-cho, Otaru 047-02, Japan,
Published online:
■ 5-(2-Nitroethynyl)salicylanilides, 6-(2-Nitroethenyl)-3-alkyl-2H-1,3-benzoxazine-2,4-dione, and Related Compounds and Their Antimicrobial and Molluscicidal Activity
N. Latif, N. S. Girgis, and F. M. Assad
*Natural Products Department, National Research Centre, Dokki, Cairo, Egypt