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HETEROCYCLES
An International Journal for Reviews and Communications in Heterocyclic ChemistryWeb Edition ISSN: 1881-0942
Published online by The Japan Institute of Heterocyclic Chemistry
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Special Issue
Special Issues of the 19th International Congress of Heterocyclic Chemistry's Special Issues, Vol. 21, No. 2, 1984
Published online:
■ A Novel Alkynylation Reaction of Epoxyalcohols
Masahiko Yamaguchi and Ichiro Hirao
*Department of Industrial Chemistry, Faculty of Engineering, Kyushu Institute of Technology, 1-1 Sensuicho, Tobata, Kitakyushu, 804-8550, Japan
Published online:
■ Synthesis of 1-Benzazocin-5-one Derivative Having Aziridine Ring
Keiichi Nomura, Makoto Takeuchi, and Katsutada Masuda
*Faculty of Pharmaceutical Sciences, Toyama Medical and Pharmaceutical University, 2630 Sugitani, Toyama, Toyama 930-0194, Japan
Published online:
■ Effective Route to Azetidines from Azetidin-2-ones with the Use of Hydroalanes as Specific Reducing Agents
Mitsuo Yamashita and Iwao Ojima
*Sagami Central Research Center, 4-4-1 Nishi-Ohnuma, Sagamihara, Kanagawa 229-0012, Japan
Published online:
■ Aluminium Chloride-catalyzed Reactions of 4-Aryl-2-chloro- and 3-Aryl-2-chlorothiophenes with Some Aromatic Compounds
T. Sone, K. Sato, and Y. Umetsu
*Department of Materials Science and Engineering, Faculty of Engineering, Yamagata University, 4-3-16 Jyonan, Yonezawa 992-8510, Japan
Published online:
■ An Investigation into the Chlorosulfonation of Acetophenone and Some Derivatives
Darek D. Chapman
*Office Imaging Research and Technology Development, Eastman Kodak Company, Rochester, New York 14650-2106, U.S.A.
Published online:
■ New Method for Syntheses of Furanone Derivatives Using Dianions
Kazuhiko Tanaka, Yutaka Isobe, Hidemi Yoda, and Aritsune Kaji
*Department of Chemistry, Faculty of Science, Kyoto University, Sakyo, Kyoto 606-8502, Japan
Published online:
■ Highly Efficient Synthesis of γ-Lactones with Titanium Homoenolates
Eiichi Nakamura, Hiroji Oshino, and Isao Kawajima
*Department of Chemistry, Faculty of Science, Tokyo Instituteof Technology, Meguro-ku, Tokyo 152-8552, Japan
Published online:
■ New Methods for the Synthesis of 3(2H)-Furanones and 2(5H)-furanones
Hiroyuki Saimoto, Seijiro Matsubara, Koichiro Oshima, Tamejiro Hiyama, and Hitosi Nozaki
*Department of Induatrial Chemistry, Faculty of Engineering, Kyoto University, Yoshida, Sakyou-ku, Kyoto 606-8501, Japan
Published online:
■ A New Method for the Synthesis of Functionalized Tetrahydrofurans and Tetrahydropyrans Directed toward the Total Synthesis of Polyether Antibiotics
Y. Oikawa, K. Horita, I. Noda, and O. Yonemitsu
*Faculty of Pharmaceutical Sciences, Hokkaido University, Kita 12 Nishi 6, Kita-ku, Sapporo, Hokkaido 060-0812, Japan
Published online:
■ Silica Gel-promoted γ-Lactonization of γ-Halo Esters
Sadao Tsuboi, Koichi Muranaka, Hiroshi Fujita, Katsuhiko Seko, and Akira Takeda
*Department of Synthetic Chemistry, Faculty of Engineering, Okayama University, 2-1-1 Tsushima-naka, Okayama 700-8530, Japan
Published online:
■ Facile Preparation of 2,6-Dimethyl-2,6-tetrahydropyrancarbolactone, a Versatile Intramediate for the Syntheses of (±)-Frontalin, (±)-Cinenic Acid, and (±)-Linaloyl Oxide
Masanori Utaka, Sadao Tsuboi, Hiroshi Makino, Yukito Oota, and Akira Takeda
*Department of Synthetic Chemistry, Faculty of Engineering, Okayama University, 2-1-1 Tsushima-naka, Okayama 700-8530, Japan
Published online:
■ Novel Synthetic Methods of Dihydro-4-pyrone, γ-Butyrolactone, and 3(2H)-Furanone by Using α,α’-Dihalo Ketone or α-Monohalo Ketone
Takashi Sakai, Mutsumi Ishikawa, Akitoshi Yamawaki, Hiroshi Ito, Eiichiro Amano, and Akira Takeda
*Department of Synthetic Chemistry, Faculty of Engineering, Okayama University, 2-1-1 Tsushima-naka, Okayama 700-8530, Japan
Published online:
■ Reaction of Methyl 12-Hydroxyabietan-8,11,13-triene-19-oate with Thallium(III) Perchlorate. Formation of a Lactone with a New Rearranged Skeleton
Tatsuhiko Nakano, María Isabel Hernández, and Andrew T. McPhail
*Centro de Química, Instituto Venezolano de Investigaciones Científicas, I.V.I.C., Apartado 21827, Caracas 1020-A, Venezuela
Published online:
■ Oxidation Reactions of Bicyclic Pyrrole Derivatives
Yoshio Otsuji, Nobuhiko Ohmura, Saburo Nakanishi, and Kazuhiko Mizuno
*Department of Applied Chemistry, College of Engineering, University of Osaka Prefecture, Sakai, Osaka 593-8531, Japan
Published online:
■ Novel Base-catalyzed 1,3-Dipolar Cycloaddition Leading to Pyrrolidines from N-(Phenylthiomethyl)amino Acids
Nobuyuki Imai, Yoshiyasu Terao, Kazuo Achiwa, and Minoru Sekiya
*Shizuoka College of Pharmacy, 2-2-1, Oshika, Shizuoka-shi, 442 Shizuoka, Japan
Published online:
■ Preparation of Optically Active Phosphonic Acid Derivatives Using Ethyl L-Prolinate and Their Application to Asymmetric Organic Synthesis
Toru Koizumi, Masanori Iwata, Nobuyuki Tanaka, Kazuhiko Hirutani, and Eiichi Yoshii
*Faculty of Pharmaceutical Sciences, Toyama Medical and Pharmaceutical University, 2630 Sugitani, Toyama, Toyama 930-0194, Japan
Published online:
■ Syntheses of Five-membered Heterocycles Containing Both Ring and Side-chain Phosphorus Atoms
Md. Amin, D. G. Holah, A. N. Hughes, and T. Rukachaisirikul
*Department of Chemistry, Lakehead University, Thunder Bay, Ontario, P7B 5E1, Canada
Published online:
■ Stereoselective Total Synthesis of Pyrrolizidine Alkaloid Bases, (-)-Rosmarinecine and (-)-Isoretronecanol
Kuniaki Tatsuta, Hideaki Takahashi, Yoshiya Amemiya, and Mitsuhiro Kinoshita
*Department of Applied Chemistry, Faculty of Science and Technology, Keio University, Hiyoshi, Kohoku-ku Yokohama 223-8522, Japan
Published online:
■ Reactions of Trifluoroacetonitrile Ylides with Electron-deficient Olefins and Acetylenes
Kiyoshi Tanaka, Hiroki Daikaku, and Keiryo Mitsuhashi
*Department of Chemistry, Faculty of Engineering, Seikei University, Musashino-shi, Tokyo 180-8633, Japan
Published online:
■ Reactivity of Isoselenazole Derivatives
Francesco Lucchesini, Vincenzo Bertini, and Angela De Munno
*Dipartimento di Chimica e Chimica Industriale, Università di Pisa, Via Risorgnimento 35, I-56126 Pisa, Italy
Published online:
■ Synthesis of Thiazoline, Thiophene, and 1,3-Dithiolane Using Ethyl 4-Haloacetoacetane
Takuo Chiba, Hirotoshi Sato, and Tetsuzo Kato
*Pharmaceutical Institute, Tohoku University, Aobayama, Sendai 980-8578, Japan
Published online:
■ C-Alkylation, Alkenylation, and Arylation of 1,2,5-Thiadiazoles
Vincenzo Bertini, Angela De Munno, and Nevio Picci
*Dipartimento di Chimica e Chimica Industriale, Università di Pisa, Via Risorgnimento 35, I-56126 Pisa, Italy
Published online:
■ A New Aromatic Annelation Reaction Utilizing Reaction of Isoxazole with Diironnonacarbonyl
Naoki Takeuchi, Kousuke Okazaki, Junji Ohki, and Seisho Tobinaga
*Showa Pharmaceutical University, 3-3165, Higashi-tamagawagakuen, Machida, Tokyo 194-8543, Japan
Published online:
■ The Mechanism of Asymmetric Transformation of 2-Substituted Alkanoic Acids
Saizo Shibata, Hajime Matsushita, Hajime Kaneko, Msao Noguchi, Masahiko Saburi, and Sadao Yoshikawa
*Central Reseasrch Institute, Japan Tobacco Inc., 6-2, Umegaoka, Midori-ku, Yokohama, Kanagawa 227-8512, Japan
Published online:
■ Diles-Alder Reaction of Oxazoles
Toshikazu Ibata and Shuji Nakano
*Department of Chemistry, Graduate School of Science, Osaka University, Toyonaka, Osaka 560-8531, Japan
Published online:
■ On the Reaction of 5-Aminoisoxazoles as Ambident Nucleophiles: Synthesis of 4,7-Dihydroisoxazolo[5,4-b]pyridines
T. Yamamori, Y. Hiramatsu, K. Sakai, and I. Adachi
*Shionogi Research Laboratories, Shionogi & Co. Ltd., Fukushima-ku, Osaka 553-0002, Japan
Published online:
■ Air Oxidation Reaction of Diazoalkenes Efficient Oxygen-transfer Reaction to Give Epoxyketones
Tsutomu Miyashi, Masaki Kamata, Yoshinori Nishizawa, and Toshio Mukai
*Department of Chemistry, Faculty of Science, Tohoku University, Aoba-ku, Ssendai 980-8578, Japan
Published online:
■ Trimethylsilyldiazomethane: A New Synthon for the Preparation of Pyrazoles
Sumie Inoue, Kimio Sudo, Toyohiko Aoyama, and Takayuki Shioiri
*Faculty of Pharmaceutical Sciences, Nagoya City University, Tanabe-dori, Mizuho-ku, Nagoya 467-8603, Japan
Published online:
■ The Selective Synthesis of Pyrazoles
Choji Kashima and Nobutoshi Yoshiwara
*Department of Chemistry, Faculty of Education, Tokyo Gakugei University, 4-1-1 Nukuikitamati, Koganei-shi, Tokyo 184, Japan
Published online:
■ Photochemistry of the Nitrogen-containing Thiocarbonyl System
Kazuaki Oda, Minoru Machida, and Yuichi Kanaoka
*Faculty of Pharmaceutical Scicences, Higashinihonngakuen University, 1757 Kanazawa, Toubetu-cho, Ishikari-gun, Hokkaodo 061-0212, Japan